EZM0414 TFA( —— )

Catalog No. M34899 CAS No. 2411759-92-5

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Get Quotation Bulk Inquiry Add to Cart

Product Name

EZM0414 TFA
Note

Research use only, not for human use.
Brief Description

EZM0414 TFA (SETD2-IN-1 TFA) is a SETD2 inhibitor with anticancer and antiproliferative effects for the study of leukemia and immune dysfunction.
Description

EZM0414 TFA is a potent, selective and orally active inhibitor of SETD2 which is a human histone methyltransferase. EZM0414 TFA has anti-proliferative effects.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

Histone Methyltransferase
Research Area

——
Indication

——

CAS Number

2411759-92-5
Formula Weight

514.51
Molecular Formula

C24H30F4N4O4
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 200 mg/mL (388.72 mM; Ultrasonic ) H2O : 6.67 mg/mL (12.96 mM; Ultrasonic (<60°C))
SMILES

OC(=O)C(F)(F)F.CC(=O)N1CCN(CC1)[C@H]1CCC[C@H](C1)NC(=O)c1cc2c(F)ccc(C)c2[nH]1
Chemical Name

——

1. John Lampe, et al. Substituted indoles and methods of use thereof. WO2020037079A1.

Calculator

molnova catalog